GlyT1


Elevation of extracellular synaptic glycine concentration by blockade of GlyT1 has been hypothesized to potentiate NMDA receptor function in vivo and to represent a rational approach for the treatment of schizophrenia and cognitive disorders.
  • VUF 11207 fumarate EI2918

    VUF 11207 fumarate是活性的 ACKR3 (CXCR7) 激动剂。

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  • SCH 51344 EI2511

    SCH 51344是活性的 MTH1 抑制剂。

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  • SB 332235 EI2480

    SB 332235是活性的 CXCR2 拮抗剂。

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  • SB 265610 EI2474

    SB 265610是活性的 CXCR2 拮抗剂。

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  • Org 24598 lithium salt EI2022

    Org 24598 lithium salt是选择性 GlyT1 抑制剂。

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